EventsThe 25th International Electronic Conference on Synthetic Organic Chemistry
Event submissions
Published
with-doi10.3390/ecsoc-25-11785
This submission belongs to the session S1. General Organic Synthesis of the event The 25th International Electronic Conference on Synthetic Organic Chemistry
Published date
14 Nov, 2021
Academic Editor
author-avatarGyörgy Keglevich
Citation
Fidel Rodríguez-López, Hugo A. García-Gutiérrez, Rocio Gámez-Montaño, Synthesis of triterpenoid-derived α-acyloxycarboxamides via Passerini reaction, in Proceedings of The 25th International Electronic Conference on Synthetic Organic Chemistry, 15 November–30 November 2021, MDPI: Basel, Switzerland, doi: 10.3390/ecsoc-25-11785
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Synthesis of triterpenoid-derived α-acyloxycarboxamides via Passerini reaction

Fidel Rodríguez-López 1
Hugo A. García-Gutiérrez 1
Rocio Gámez-Montaño 2
1. Instituto de Investigaciones Químico Biológicas, Universidad Michoacana de San Nicolás de Hidalgo
2. Departamento de Química, Universidad de Guanajuato
Abstract

Herein we describe the synthesis of a small series of α-acyloxycarboxamides via a facile and efficient one-pot procedure, employing a plant-derived triterpenoid as carboxylic acid component. The products were obtained in overall yields of 25 to 79%, while we scoped the effect of the nature of the aldehyde component on the reaction yields.

Keywords
Passerini reaction (P-3CR)
α-acyloxycarboxamides
triterpenoid
Manuscript
sciforum-051652ECSOC 21 FRL_7.pdf
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