Events8th International Electronic Conference on Medicinal Chemistry
Published
with-doi10.3390/ECMC2022-13408 (registering DOI)
This submission belongs to the session S3. General of the event 8th International Electronic Conference on Medicinal Chemistry
Published date
01 Nov, 2022
Academic Editor
author-avatarAlfredo Berzal-Herranz
Citation
Salvatore Princiotto, Stefania Mazzini, Loana Musso, Roberto Artali, Raimundo Gargallo, Anna Aviñó, Ramon Eritja, Vera Isca, Sabrina Dallavalle, Evaluation of the interactions of selected ligands with (3+1) G-quadruplex sequence within PARP1 gene promoter region, in Proceedings of 8th International Electronic Conference on Medicinal Chemistry, 1 November–30 November 2022, MDPI: Basel, Switzerland, doi: 10.3390/ECMC2022-13408
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Evaluation of the interactions of selected ligands with (3+1) G-quadruplex sequence within PARP1 gene promoter region

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1. Department of Food, Environmental and Nutritional Sciences (DEFENS), University of Milan, via Celoria, 2, 20133 Milan, Italy
2. Universidade Lusófona de Humanidades e Tecnologias, Escola de Ciências e Tecnologias da Saúde, Campo Grande 376, 1749-024 Lisboa
3. University of Milan, Department of Food, Environmental and Nutritional Sciences (DEFENS), Via G. Celoria 2, 20133 Milan, Italy
4. Scientia Advice di Roberto Artali, 20832 Desio, Milan, Italy
5. Universidade Lusófona de Humanidades e Tecnologias, Escola de Ciências e Tecnologias da Saúde, Campo Grande 376, 1749-024 Lisboa, Portugal
6. Institute for Advanced Chemistry of Catalonia (IQAC), CSIC, Networking Center on Bioengineering, Biomaterials and Nanomedicine (CIBER-BBN), c/ Jordi Girona 18-26, 08034 Barcelona, Spain
7. University of Barcelona, Department of Chemical Engineering and Analytical Chemistry, Martí i Franquès, 1-11, 08028 Barcelona, Spain
Abstract
Keywords
G-quadruplex
PARP
hybrid
ligand
interaction
stabilization