This submission belongs to the session a. General Organic Synthesis of the event The 10th International Electronic Conference on Synthetic Organic Chemistry
Published date
30 Nov, 2006
Citation
Jeanne-Marie Begouin, Stéphanie Hesse, Synthesis of novel benzoannelated eight-membered heterocycles: easy access to benzo[f][1,4]oxazocin-1-ones, in Proceedings of The 10th International Electronic Conference on Synthetic Organic Chemistry, 1 November–30 November 2006, MDPI: Basel, Switzerland, doi: 10.3390/ecsoc-10-01384
Share
Email
Facebook
Twitter
LinkedIn
Synthesis of novel benzoannelated eight-membered heterocycles: easy access to benzo[f][1,4]oxazocin-1-ones
Jeanne-Marie Begouin 1
Stéphanie Hesse 1
1. Laboratoire d’Ingénierie Moléculaire et Biochimie Pharmacologique, Université Paul Verlaine - Metz, 1 Boulevard Arago, 57070 METZ, France
Abstract
Medium-sized N-heterocycles, in particular eight-membered azocines, are key structures occurring in many natural products and in some compounds having biological activities. We described here an easy access to benzo[f][1,4]oxazocin-1-ones starting from 2-acetylbenzoic acid.
Keywords
eight-membered N
O heterocycles
ethanolamines
ZnCl<sub>2</sub>
Reaction of azaheterylguanidines with trichloroacetonitrile
Synthesis of Cyclic Enehydrazides by Ring-Closure Metathesis. Application to the Enantioselective Synthesis of 2-Alkyl and Aryl Piperidines