Event submissions
Published
This submission belongs to the session S3. Immune and Inflammatory Diseases of the event The 1st International Online Conference on Diseases
Published date
05 Sep, 2025
Academic Editor
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Veysel TahanCitation
Ekaterina Dmitrievna Savina, Ekaterina Mikhailovna Zhidkova, Daria Vladimirovna Stepanycheva, Pavel Aleksandrovich Kusov, Kirill Vladimirovich Gordeev, Andrey Valerievich Matveev, Marianna Gennadievna Yakubovskaya, Ekaterina Andreevna Lesovaya, Anti-cancer activity of novel selective glucocorticoid receptor agonist 13S-G2 in vitro on the model of blood cancer, in Proceedings of The 1st International Online Conference on Diseases, 9 September–11 September 2025, MDPI: Basel, Switzerland
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Anti-cancer activity of novel selective glucocorticoid receptor agonist 13S-G2 in vitro on the model of blood cancer
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Ekaterina Dmitrievna Savina 1
Ekaterina Mikhailovna Zhidkova 1
Daria Vladimirovna Stepanycheva 1
Pavel Aleksandrovich Kusov 2
Kirill Vladimirovich Gordeev 3
Andrey Valerievich Matveev 4
Marianna Gennadievna Yakubovskaya 1,5
Ekaterina Andreevna Lesovaya 1,5,6
1. Department of Chemical Carcinogenesis, Institute of Carcinogenesis, N.N. Blokhin National Medical Research Center for Oncology, Kashirskoe Shosse 24-15, Moscow 115478, Russia
2. Independent researcher, Moscow, Russia
3. Faculty of Pharmacy, Kuban State Medical University, Ministry of Health of Russia, 4 Mitrofan Sedin Str., Krasnodar 350063, Russia
4. Department of Biotechnology and Industrial Pharmacy, Lomonosov Institute of Fine Chemical Technologies, MIREA—Russian Technological University, 86 Vernadsky Prospekt, Moscow 119571, Russia
5. Institute of Medicine, Peoples’ Friendship University of Russia, Miklukho-Maklaya St. 6, Moscow 117198, Russia
6. Faculty of Oncology, I.P. Pavlov Ryazan State Medical University, Vysokovol’tnaya Str. 9, Ryazan 390026, Russia
Abstract
Keywords
glucocorticoids
glucocorticoid receptor
selective glucocorticoid receptor agonist
synephrine
hematological malignancies
transrepression
transactivation