This submission belongs to the session b. Bioorganic, Medicinal and Natural Products of the event The 15th International Electronic Conference on Synthetic Organic Chemistry
Published date
27 Oct, 2011
Citation
Josef Jampilek, Katarina Kralova, Pavel Bobal, Jiri Kos, Tomas Gonec, Matus Pesko, Josef Sujan, Preparation and Herbicidal Properties of Substituted Quinoline-2-carboxanilides, in Proceedings of The 15th International Electronic Conference on Synthetic Organic Chemistry, 1 November–30 November 2011, MDPI: Basel, Switzerland, doi: 10.3390/ecsoc-15-00588
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Preparation and Herbicidal Properties of Substituted Quinoline-2-carboxanilides
Josef Jampilek 1
Katarina Kralova 2
Pavel Bobal 1
Jiri Kos 1
Tomas Gonec 1
Matus Pesko 3
Josef Sujan 1
1. Department of Chemical Drugs, Faculty of Pharmacy, University of Veterinary and Pharmaceutical Sciences
2. Institute of Chemistry, Faculty of Natural Sciences, Comenius University
3. Department of Ecosozology and Physiotactics, Faculty of Natural Sciences, Comenius University
Abstract
In this study a series of twenty-five substituted quinoline-2-carboxanilides were prepared. The procedures for synthesis of the compounds are presented. The compounds were tested for their activity related to inhibition of photosynthetic electron transport (PET) in spinach (Spinacia oleracea L.) chloroplasts. For all the compounds the structure-activity relationships (SAR) are discussed.
Keywords
quinoline-2-carboxanilides
PET inhibition
spinach chloroplasts
structure-activity relationships
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