Events6th International Electronic Conference on Medicinal Chemistry
Published
This submission belongs to the session H. Round Table on Parasitic Diseases of the event 6th International Electronic Conference on Medicinal Chemistry
Published date
06 Nov, 2020
Citation
Melanie Fonte, Natália Tassi, Diana Fontinha, Inés Bouzón-Arnáiz, Ricardo Ferraz, Maria J. Araújo, Xavier Fernàndez-Busquets, Miguel Prudêncio, Paula Gomes, Cátia Teixeira, 4,9-Diaminoacridines and 4-aminoacridines as antiplasmodial dual-stage hits, in Proceedings of 6th International Electronic Conference on Medicinal Chemistry, 1 November–30 November 2020, MDPI: Basel, Switzerland, doi: 10.3390/ECMC2020-07493
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4,9-Diaminoacridines and 4-aminoacridines as antiplasmodial dual-stage hits

Inés Bouzón-Arnáiz 4,5
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Maria J. Araújo 2
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1. LAQV-REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Portugal.
2. LAQV-REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Portugal
3. Instituto de Medicina Molecular, Faculdade de Medicina, Universidade de Lisboa, Portugal
4. Nanomalaria Group, Institute for Bioengineering of Catalonia (IBEC), The Barcelona Institute of Science and Technology, Spain
5. Barcelona Institute for Global Health (ISGlobal), Barcelona Center for International Health Research (CRESIB), Hospital Clínic-Universitat de Barcelona, Spain
6. Ciências Químicas e das Biomoléculas, Escola Superior de Saúde, Politécnico do Porto, Portugal
7. Nanoscience and Nanotechnology Institute (IN2UB), University of Barcelona, Spain
Abstract
Keywords
acridines
antimalarial activity
blood-stage
liver-stage
multi-target drugs
organic synthesis