In recent years, herbal medicines have garnered worldwide attention from both people and researchers due to their aesthetic value, improved patient compliance, and significant therapeutic effects. Herbal drugs can be more effectively utilized by incorporating them into modern dosage forms. This can be achieved through the design of novel herbal ingredient drug delivery systems, which represent innovative approaches addressing the limitations of traditional drug delivery systems. Implementing novel drug delivery technologies in herbal medicine has the potential to enhance efficacy and reduce the side effects associated with various herbal compounds and herbs.These formulations offer several advantages over traditional methods, including improved solubility and bioavailability, reduced toxicity, controlled drug delivery, and protection of plant actives from degradation. Moreover, they exhibit drug-targeting properties that enhance selectivity, delivery precision, and overall effectiveness, often allowing for dose reduction. These advancements not only increase safety but also promote patient compliance.Various novel herbal drug delivery systems include liposomes, phytosomes, nanoemulsions, nanoparticles, ethosomes, and transferosomes, each offering unique benefits. For instance, liposomes and nanoparticles can encapsulate poorly water-soluble herbal extracts, enhancing their absorption and stability. Phytosomes improve the bioavailability of polyphenolic compounds, while nanoemulsions enhance skin penetration in topical applications. These systems not only protect active constituents from environmental degradation but also improve therapeutic indices by ensuring site-specific delivery.Furthermore, these technologies can be applied to both traditional herbal formulations and modern herbal products, bridging the gap between conventional herbal therapy and advanced pharmaceutical science. With continued research and development, novel herbal drug delivery systems are poised to revolutionize the way herbal medicines are administered, making them safer, more effective, and more acceptable to modern consumers.